02:49CYP Activity Quantification in Cell Cultures: Metabolic Probes, Inducers, and Inhibitors
04:30CYP Activity Quantification in Cell Cultures: Medium Treatment
05:40CYP Activity Quantification in Cell Cultures: Mass Spectrometry (MS)-based Quantification
06:49CYP Activity Quantification in Cell Cultures: Probes Using Luminescence-based Methods
08:10Results: Quantification of Metabolites Produced by tha Activity of CYP Enzymes Following Cell Incubation with CYP Inducers, Substrates, and Inhibitors
Competenza metabolica dei sistemi in vitro è un requisito fondamentale per la biotrasformazione e la disposizione di farmaci e sostanze tossiche. In questo protocollo, si descrive l'applicazione di sonde metabolici riferimento per valutare fase del metabolismo in colture cellulari.